Beilstein J. Org. Chem.2020,16, 982–988, doi:10.3762/bjoc.16.87
thus be rapidly accessed, identifying privileged or challenging scaffolds and paving the way for further exploration.
Keywords: benchtopanalytics; fragment-based library; heterocyclic sp2–sp3 fragments; N-arylation; photoredox-nickel dual catalysis; Introduction
Heterocyclic sp2–sp3 fragments are